{"id":34,"date":"2017-08-02T11:42:58","date_gmt":"2017-08-02T11:42:58","guid":{"rendered":"http:\/\/www.tsklifesciences.com\/?page_id=34"},"modified":"2023-05-06T03:18:47","modified_gmt":"2023-05-06T03:18:47","slug":"intermediates","status":"publish","type":"page","link":"https:\/\/www.tsklifesciences.com\/?page_id=34","title":{"rendered":"INTERMEDIATES"},"content":{"rendered":"<style type=\"text\/css\">\n<!-- .style3 {color: #FFFFFF; font-weight: bold; } --><br \/><\/style>\n<table border=\"0\" width=\"100%\" cellspacing=\"1\" cellpadding=\"0\">\n<tbody>\n<tr>\n<td valign=\"middle\" bgcolor=\"0066CC\" height=\"35\">\n<p class=\"style3\" align=\"center\">Name of the Intermediate<\/p>\n<\/td>\n<td valign=\"middle\" bgcolor=\"0066CC\" height=\"35\">\n<p class=\"style3\" align=\"center\">CAS<\/p>\n<\/td>\n<td valign=\"middle\" bgcolor=\"0066CC\" height=\"35\">\n<p class=\"style3\" align=\"center\">Application \/API Name<\/p>\n<\/td>\n<td valign=\"middle\" bgcolor=\"0066CC\" height=\"35\">\n<p class=\"style3\" align=\"center\">Production status<\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>3,4-Dihydroxybenzaldehyde<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>139-85-5<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Roflumilast\/ Fine chemical<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial <\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2,4-dimethyl-benzenethiol<\/strong><br \/>\n<strong>2,4-dimethyl thiophenol<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>13616-82-5<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Vortioxetine<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>(2,4-dimethylphenyl)(2-nitrophenyl)sulfane<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>1610527-49-5<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Vortioxetine<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Moc-L-Valine.<\/strong><br \/>\n<strong>(S)-2-((Methoxycarbonyl)aMino)-3-Methylbutanoic acid.<\/strong><br \/>\n<strong>N-(Methoxycarbonyl)-L-valine<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>74761-42-5<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Fine chemical<\/strong><br \/>\n<strong>Ravidasvir<\/strong><br \/>\n<strong>Daclatasvir, <\/strong><br \/>\n<strong>\u00a0Ledipasvir<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>L-Valine methyl ester hydrochloride<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>6306-52-1<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Fine chemical<\/strong><br \/>\n<strong>Valsartan<\/strong><br \/>\n<strong>Ritonavir<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>5,6-Dimethoxy -1-indanone<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2107-69-9<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Donepezil<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>5-Bromo-6-methoxy-1-indanone<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>187872-11-3<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Advanced intermediate<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pilot Scale<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>1-phenyl-1,2,3,4-tetrahydroisoquinoline<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>22990-19-8<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Solifenacin succinate<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>N-[[N-Methyl-N-[(2-isopropyl]-4-thiazolyl)methyl)amino]carbonyl-L-valine Methyl Ester <\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>154248-99-4<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Ritonavir<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>N-Carbobenzyloxy-L-valine<\/strong><br \/>\n<strong>CBZ-L-Valine<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>1149-26-4<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Valaciclovir<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>4-Amino -2- chloro-6,7- di methoxy quinazoline<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>23680-84-4<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Alfuzosin\/Terazosin\/Prazosin\/Bunazosin\/Doxazosin<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2-Chloro-4,6-dimethoxy-1,3,5-triazine (CDMT)<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>3140-73-6<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pemetrexed, peptide coupling agent<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>5-Bromo-2-chlorobenzoic acid<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>21739-92-4<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Dapagliflozin ,Empagliflozin,Bexagliflozin<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2-Chloro-5-iodobenzoic Acid<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>19094-56-5<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Dapagliflozin ,Empagliflozin,Bexagliflozin<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pilot scale<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2-Bromo-5-hydroxybenzaldehyde<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2973-80-0<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Crisaborole<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pilot scale<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Methyl carbazate,<\/strong><br \/>\n<strong>Methyl hydrazinecarboxylate<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>6294-89-9<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Aprepitant<\/strong><br \/>\n<strong>Nefazodone hydrochloride<\/strong><br \/>\n<strong>Fine chemical<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Isobutyramide<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>563-83-7<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Fine chemical\/<\/strong><br \/>\n<strong>Ritonavir<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Commercial<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>5-amino-2-chloro-4-fluorophenol<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>84478-72-8<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Advanced intermediate<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pilot Scale<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>3-amino-4-fluorophenol<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>62257-16-3<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Advanced intermediate<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pilot Scale<\/strong><\/p>\n<\/td>\n<\/tr>\n<tr>\n<td valign=\"middle\">\n<p align=\"center\"><strong>2-Chloro-4-fluorophenol<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>1996-41-4\u00a0 <\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Advanced intermediate<\/strong><\/p>\n<\/td>\n<td valign=\"middle\">\n<p align=\"center\"><strong>Pilot Scale<\/strong><\/p>\n<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p><strong>Note :<\/strong> All Transactions are carried out in conformity with the patent laws applicable in the user country. Responsibility with respect to third party\u2019s patent rights in a specific country lies exclusively with the buyer.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Name of the Intermediate CAS Application \/API Name Production status 3,4-Dihydroxybenzaldehyde 139-85-5 Roflumilast\/ Fine chemical Commercial 2,4-dimethyl-benzenethiol 2,4-dimethyl thiophenol 13616-82-5 Vortioxetine Commercial (2,4-dimethylphenyl)(2-nitrophenyl)sulfane 1610527-49-5 Vortioxetine Commercial Moc-L-Valine. (S)-2-((Methoxycarbonyl)aMino)-3-Methylbutanoic acid. N-(Methoxycarbonyl)-L-valine 74761-42-5 Fine chemical Ravidasvir Daclatasvir, \u00a0Ledipasvir Commercial L-Valine methyl ester hydrochloride 6306-52-1 Fine chemical Valsartan Ritonavir Commercial 5,6-Dimethoxy -1-indanone 2107-69-9 Donepezil Commercial 5-Bromo-6-methoxy-1-indanone 187872-11-3 Advanced&hellip;<\/p>\n<p class=\"more-link\"><a href=\"https:\/\/www.tsklifesciences.com\/?page_id=34\" class=\"themebutton2\">Read More<\/a><\/p>\n","protected":false},"author":1,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":{"footnotes":""},"class_list":["post-34","page","type-page","status-publish","hentry"],"_links":{"self":[{"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=\/wp\/v2\/pages\/34","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=34"}],"version-history":[{"count":9,"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=\/wp\/v2\/pages\/34\/revisions"}],"predecessor-version":[{"id":193,"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=\/wp\/v2\/pages\/34\/revisions\/193"}],"wp:attachment":[{"href":"https:\/\/www.tsklifesciences.com\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=34"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}